To synthesize new derivatives of quinazolinones by the Buchwald-Hartwig method, 6-bromo-quinazolin-4-one derivatives were initially synthesized using cyclization methods and converted into 6-bromoquinazolin-4-thiones using Lawesson's reagent. These thione derivatives were reacted with aromatic amines in the presence of appropriate bases, palladium catalysts, and solvents, their chemical properties were studied and optimal conditions were selected. The structures of the resulting new compounds were studied based on 1H NMR, 13C NMR, MS, and MP analyses.
| Mualliflar | Davron Turgunov, Azizbek Nasrullaev, Khurshed Bozorov, N. Lifei, Haji Akber Aisa |
|---|---|
| Jurnal | Samarqand davlat universiteti ilmiy tadqiqotlar axborotnomasi |
| Nashriyot | Самарқанд давлат университети |
| ISSN | 2091-5446, 2181-1296 |
| Nashr sanasi | 2025-03-29 |
| Jild | 1 |
| Son | 1 |
| Betlar | 23-28 |
| Til | Ingliz |
| Ilmiy soha | Kimyo |
| DOI | 10.59251/2181-1296.2025.v1.149.2.3210 |
| Indeksga qo‘shilgan | 2026-09-02 |
DOI: 10.59251/2181-1296.2025.v1.149.2.3210 · Maqolaning asl sahifasi
| APA | Davron Turgunov, Azizbek Nasrullaev, Khurshed Bozorov, N. Lifei, & Haji Akber Aisa (2025). SYNTHESIS OF 6-SUBSTITUTED QUINAZOLINE-4-THIONES BY THE BUCHWALD HARTWIG METHOD. Samarqand davlat universiteti ilmiy tadqiqotlar axborotnomasi, 1(1), 23-28. https://doi.org/10.59251/2181-1296.2025.v1.149.2.3210 |
|---|---|
| GOST (OAK) | Davron Turgunov va b. SYNTHESIS OF 6-SUBSTITUTED QUINAZOLINE-4-THIONES BY THE BUCHWALD HARTWIG METHOD // Samarqand davlat universiteti ilmiy tadqiqotlar axborotnomasi. – 2025. – T. 1, № 1. – P. 23-28. – DOI: 10.59251/2181-1296.2025.v1.149.2.3210. |
| MLA | Davron Turgunov, Azizbek Nasrullaev, Khurshed Bozorov, N. Lifei, and Haji Akber Aisa. “SYNTHESIS OF 6-SUBSTITUTED QUINAZOLINE-4-THIONES BY THE BUCHWALD HARTWIG METHOD.” Samarqand davlat universiteti ilmiy tadqiqotlar axborotnomasi, 1(1), 23-28, 2025. https://doi.org/10.59251/2181-1296.2025.v1.149.2.3210 |
| Chicago | Davron Turgunov, Azizbek Nasrullaev, Khurshed Bozorov, N. Lifei, and Haji Akber Aisa. “SYNTHESIS OF 6-SUBSTITUTED QUINAZOLINE-4-THIONES BY THE BUCHWALD HARTWIG METHOD.” Samarqand davlat universiteti ilmiy tadqiqotlar axborotnomasi, 1(1), 23-28 (2025). https://doi.org/10.59251/2181-1296.2025.v1.149.2.3210 |
| Harvard | Davron Turgunov, Azizbek Nasrullaev, Khurshed Bozorov, N. Lifei, and Haji Akber Aisa (2025) ‘SYNTHESIS OF 6-SUBSTITUTED QUINAZOLINE-4-THIONES BY THE BUCHWALD HARTWIG METHOD’, Samarqand davlat universiteti ilmiy tadqiqotlar axborotnomasi, 1(1), 23-28. https://doi.org/10.59251/2181-1296.2025.v1.149.2.3210 |
| BibTeX | @article{davronturgunov2025,
title = {SYNTHESIS OF 6-SUBSTITUTED QUINAZOLINE-4-THIONES BY THE BUCHWALD HARTWIG METHOD},
author = {Davron Turgunov and Azizbek Nasrullaev and Khurshed Bozorov and N. Lifei and Haji Akber Aisa},
journal = {Samarqand davlat universiteti ilmiy tadqiqotlar axborotnomasi},
year = {2025},
volume = {1},
number = {1},
pages = {23-28},
doi = {10.59251/2181-1296.2025.v1.149.2.3210},
url = {https://doi.org/10.59251/2181-1296.2025.v1.149.2.3210}
} |
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